Lub hauv paus pob txha ntawm cov tshuaj tua kab mob quinolone muaj cov qauv nitrogen (hetero) biparacyclic. Quinolone thiab lwm yam tshuaj tua kab mob muaj cov ntsiab lus sib txawv ntawm kev nqis tes ua.
Lawv tsom cov kab mob DNA (DNA). Qhov ob-kab DNA ntawm cov kab mob tau sib tw ua cov maggot lossis kauv (hu ua supercoil).
Cov enzyme uas ua DNA rau hauv supercoil hu ua DNA gyrase. Quinolones cuam tshuam cov enzyme no thiab ntxiv ua rau tsis tuaj yeem ua puas rau cov kab mob DNA. Cov hlwb tsis faib ntxiv lawm.
Lawv qhia pom cov tshuaj lom rau cov kab mob. Tam sim no, qhov tsis kam ntawm qee cov kab mob rau ntau yam tshuaj tua kab mob tuaj yeem nthuav dav vim yog kis plasmid.
Cov tshuaj hauv chav kawm no tsis cuam tshuam los ntawm plasmid-kis tsis kam, yog li tsis muaj kev tiv thaiv kab mob sib kis ntawm cov tshuaj no thiab ntau yam tshuaj tua kab mob.
B. Zoo qhov ncauj nqus thiab nthuav dav hauv lub cev. Cov ntshav protein khi rau tus nqi qis thiab ntshav ib nrab lub neej yog qhov ntev. Ib nrab raug tso tawm hauv ob lub raum, tso zis siab ntau, thiab ib feem metabolized los ntawm lub siab.
C. Tsawg qhov tsis zoo thiab zam tau zoo. Xeev siab, ntuav, tsis qab los noj mov, ua pob, mob taub hau, thiab kiv taub hau yog ib txwm muaj. Qee zaum ntuav thiab lwm yam kev mob hlwb, kev tshem tawm tuaj yeem txo qis. Txhua yam fluoroquinolones yuav tsum tsis txhob siv rau cov menyuam ua ntej pubertal lossis poj niam cev xeeb tub vim tias lawv tuaj yeem ua rau mob caj dab hauv cov menyuam yaus thiab ua rau mob sib koom thiab ua rau me nyuam yaus.
D. Tsim nyog rau cov kab mob rhiab (xws li Staphylococcus aureus, Pseudomonas aeruginosa, plab hnyuv gram-negative bacilli, Campylobacter thiab Neisseria gonorrhoeae, thiab lwm yam) paub tias muaj kab mob tso zis, mob prostate, kab mob gonorrhea, kab mob ua pa, mob plab hnyuv thiab kis kab mob hauv pob txha, pob qij txha, thiab cov nqaij mos.
Kev siv Quinolones
1. Quinolone pob ntseg poob
Ofloxacin pob ntseg poob, qhov taw qhia yog rau kev kho mob ntawm otitis media, sab nrauv pob ntseg hnov pob ntseg, thiab tympanitis tshwm sim los ntawm cov kab mob rhiab.
Ofloxacin yog cov tshuaj tua kab mob, uas ua rau A subunit ntawm cov kab mob DNA helicase, txwv tsis pub DNA sib txuas thiab rov ua dua thiab ua rau cov kab mob tuag.
2. Cov tshuaj tua kab mob Quinolones
Cov tshuaj tua kab mob Quinolone yog cov tswv cuab ntawm ntau cov tshuaj tua kab uas nthuav dav uas sib koom cov qauv txheej txheem bicyclic cuam tshuam nrog 4-quinolone tshuaj. Lawv tau siv hauv tib neeg thiab tsiaj kho tsiaj los kho cov kab mob sib kis nrog rau kev ua tsiaj txhu.
Quinolones Test (0.5PPB) cov khoom siv los ntawm BALLYA tuaj yeem tshawb pom qhov muaj Quinolones seem hauv cov khoom lag luam ua liaj ua teb.
Cov khoom siv no tsis yog siv yooj yim xwb, tab sis kuj muaj lub sijhawm sim luv thiab raug qhov tseeb, thiab cov txiaj ntsig kev xeem ua raws EU qauv. Muaj peev xwm ua kom muaj kev nyab xeeb ntawm cov khoom lag luam ua liaj ua teb.
Yuav ua li cas xaj Quinolones Test?
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